You can find more information about
GCN5
using the following links:
PFID
PFID Old
Formal Annotation
PlasmoDB
TDR Targets
Subcellular Localization
Affecting Drugs
Drug Name
PubMed Articles (year of publication)
PF3D7_0823300
PF08_0034
histone acetyltransferase GCN5
PlasmoDB
TDR
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(2S)-2-[[2-fluoro-4-[(3-methyl-1-oxo-4Hbenzo[f]quinazolin-9-yl) methylamino] benzoyl]amino] pentanedioic acid
Designing novel inhibitors against histone acetyltransferase (HAT: GCN5) of Plasmodium falciparum
2-[[4-[(2-amino-4-oxo-1H-quin azolin-6-yl) methyl-(cyanometh yl)amino]benzoyl]amino] pentnedioic acid(ZINC29250560)
Designing novel inhibitors against histone acetyltransferase (HAT: GCN5) of Plasmodium falciparum
3-chloro-4-methylaniline
Arbitrarily Accessible 3D Microfluidic Device for Combinatorial High-Throughput Drug Screening
6-[4-methyl-2-oxo-5-phenylmet hoxycarbonyl- 6-(4-phenylphen yl)-1,6-dihydropyrimidin-3-yl] hexanoic acid
Designing novel inhibitors against histone acetyltransferase (HAT: GCN5) of Plasmodium falciparum
Anacardic acid
Histone acetyltransferase inhibitor anacardic acid causes changes in global gene expression during in vitro Plasmodium falciparum development
Curcumin
Cytotoxic effect of curcumin on malaria parasite Plasmodium falciparum: inhibition of histone acetylation and generation of reactive oxygen species
Synthesis and exploration of novel curcumin analogues as anti-malarial agents
Arbitrarily Accessible 3D Microfluidic Device for Combinatorial High-Throughput Drug Screening
fosmidomycin
Histone H3K9 acetylation level modulates gene expression and may affect parasite growth in human malaria parasite Plasmodium falciparum
Hybrid 4-aminoquinoline-1,3,5-triazine
Formulation of nanotized curcumin and demonstration of its antimalarial efficacy
N-[(4-amino-2-methylpyrimidin-5-yl)methyl]-N-[(Z)-5-hydroxy-3-[3-(4-methylphenyl)-3-oxopropyl]sulfanylpent-2-en-2-yl]formamide;hydrochloride
Arbitrarily Accessible 3D Microfluidic Device for Combinatorial High-Throughput Drug Screening
triazolophthalazine
Activity of bromodomain protein inhibitors/binders against asexual-stage Plasmodium falciparum parasites
Expasy - NiceZime View
Brenda - The Comprehensive Enzyme Information System