You can find more information about
multidrug resistance protein 1. MDR1, IP3 receptor
using the following links:
PFID
PFID Old
Formal Annotation
PlasmoDB
TDR Targets
Subcellular Localization
Affecting Drugs
Drug Name
PubMed Articles (year of publication)
PF3D7_0523000
PFE1150w
multidrug resistance protein 1. MDR1, IP3 receptor
PlasmoDB
TDR
Picture 1
Picture 2
2,5-diaminobenzophenone
Antimalarial and antitrypanosomal activity of a series of amide and sulfonamide derivatives of a 2,5-diaminobenzophenone
ACT-451840
CRISPR-Cas9-modified pfmdr1 protects Plasmodium falciparum asexual blood stages and gametocytes against a class of piperazine-containing compounds but potentiates artemisinin-based combination therapy partner drugs
amaranth
The Potential of Secondary Metabolites from Plants as Drugs or Leads against Protozoan Neglected Diseases-Part III: In-Silico Molecular Docking Investigations.
carmoisine
The Potential of Secondary Metabolites from Plants as Drugs or Leads against Protozoan Neglected Diseases-Part III: In-Silico Molecular Docking Investigations.
Chembl2387271
UV-triggered affinity capture identifies interactions between the Plasmodium falciparum multidrug resistance protein 1 (PfMDR1) and antimalarial agents in live parasitized cells
Chloroquine
Purified Plasmodium falciparum multi-drug resistance protein (PfMDR 1) binds a high affinity chloroquine analogue
PfMDR1: mechanisms of transport modulation by functional polymorphisms
Monitoring PfMDR1 transport in Plasmodium falciparum
Chlorpheniramine
Chemosensitization potential of P-glycoprotein inhibitors in malaria parasites
Cyclosporin a
Genetic linkage of pfmdr1 with food vacuolar solute import in Plasmodium falciparum
cyclosporin A
Influence of the Plasmodium falciparum P-glycoprotein homologue 1 (pfmdr1 gene product) on the antimalarial action of cyclosporin
Dihydroartemisinin
Monitoring PfMDR1 transport in Plasmodium falciparum
Doxycycline
PftetQ and pfmdt copy numbers as predictive molecular markers of decreased ex vivo doxycycline susceptibility in imported Plasmodium falciparum malaria
Mefloquine
Purified Plasmodium falciparum multi-drug resistance protein (PfMDR 1) binds a high affinity chloroquine analogue
PfMDR1: mechanisms of transport modulation by functional polymorphisms
Monitoring PfMDR1 transport in Plasmodium falciparum
Mk571
A 2-amino quinoline, 5-(3-(2-(7-chloroquinolin-2-yl)ethenyl)phenyl)-8-dimethylcarbamyl-4,6-dithiaoctanoic acid, interacts with PfMDR1 and inhibits its drug transport in Plasmodium falciparum
Ont-093
Genetic linkage of pfmdr1 with food vacuolar solute import in Plasmodium falciparum
P-loop ntpase, no human ortholog, suggested target
A systematic classification of Plasmodium falciparum P-loop NTPases: structural and functional correlation
polycyclic amines
Polycyclic amines as chloroquine resistance modulating agents in Plasmodium falciparum
Quinacrine
Monitoring PfMDR1 transport in Plasmodium falciparum
Quinine
Purified Plasmodium falciparum multi-drug resistance protein (PfMDR 1) binds a high affinity chloroquine analogue
PfMDR1: mechanisms of transport modulation by functional polymorphisms
Monitoring PfMDR1 transport in Plasmodium falciparum
tartazine
The Potential of Secondary Metabolites from Plants as Drugs or Leads against Protozoan Neglected Diseases-Part III: In-Silico Molecular Docking Investigations.
Verapamil
Genetic linkage of pfmdr1 with food vacuolar solute import in Plasmodium falciparum
Monitoring PfMDR1 transport in Plasmodium falciparum
Xr-9576
Genetic linkage of pfmdr1 with food vacuolar solute import in Plasmodium falciparum
Expasy - NiceZime View
Brenda - The Comprehensive Enzyme Information System