You can find more information about
multidrug resistance-associated protein 1 MRP1
using the following links:
PFID
PFID Old
Formal Annotation
PlasmoDB
TDR Targets
Subcellular Localization
Affecting Drugs
Drug Name
PubMed Articles (year of publication)
PF3D7_0112200
PFA0590w
multidrug resistance-associated protein 1 MRP1
PlasmoDB
TDR
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16α-bromoepiandrosterone
16alpha-bromoepiandrosterone, an antimalarial analogue of the hormone dehydroepiandrosterone, enhances phagocytosis of ring stage parasitized erythrocytes: a novel mechanism for antimalarial activity
2,3-dimethylbutyl N-(4-(((benzyloxy)carbonyl)amino)-5-(((3-methylbutan-2-yl)oxy)methyl)hex-5-enoyl)-S-(2,4-dinitrophenyl)cysteinylglycinate
Antimicrobial effects of N-benzyloxycarbonyl-S-(2,4-dinitrophenyl) glutathione diesters against chloroquinine sensitive (NF54) and resistant (K1) strains of Plasmodium falciparum
2-[[(1-Amino-4-phenylbutyl)hydroxyphosphinyl]-methyl]-3-(4-hydroxyphenyl)propionic Acid
A chemical proteomics approach for the search of pharmacological targets of the antimalarial clinical candidate albitiazolium in Plasmodium falciparum using photocrosslinking and click chemistry
Dantrolene
Glutathione export from human erythrocytes and Plasmodium falciparum malaria parasites
Furosemide
Glutathione export from human erythrocytes and Plasmodium falciparum malaria parasites
Isg-21
Glutathione export from human erythrocytes and Plasmodium falciparum malaria parasites
Mk571
Glutathione export from human erythrocytes and Plasmodium falciparum malaria parasites
Quinine
Polymorphisms within PfMDR1 alter the substrate specificity for anti-malarial drugs in Plasmodium falciparum
Substrate specificity, mutations, suggested target
Disruption of a Plasmodium falciparum multidrug resistance-associated protein (PfMRP) alters its fitness and transport of antimalarial drugs and glutathione
Tp-52
Glutathione export from human erythrocytes and Plasmodium falciparum malaria parasites
Expasy - NiceZime View
Brenda - The Comprehensive Enzyme Information System