You can find more information about chloroquine resistance transporter using the following links:

PlasmoDB - the Plasmodium genome resource
The TDR Targets Database

Subcellular Localization

PDB protein strucure

Affecting Drugs
Drug Name PubMed Articles (year of publication)
1,4-dimethoxynaphthalene
1,4-naphthoquinone
3-chloro-6-(2-diethylamino-ethoxy)-10-(2-diethylamino-ethyl)-acridone
4-amino-7-chloroquinolines
4-aminoquinoline
9,10-dihydroethanoanthracene derivatives
acridine orange
amantadine
Amodiaquine
Artemisinin
Benzoxazine
Blasticidin s
Brefeldin a
Chloroquine
Chlorpheniramine
Cinchona stereoisomer pairs: quinine and quinidine; cinchonidine and cinchonine; hydroquinine and hydroquinidine; 9-epiquinine and 9-epiquinidine
Desipramine
Dibemethin
Dynasore
Ferroquine
Fluoxetine
Hemoglobin digestion
Methylene blue
Morpholino oligomer
N-((3-Chlorophenyl)(4-(piperazin-1-ylmethyl)phenyl)methyl)-5-methoxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
N-(3-((7-chloroquinolin-4-yl)amino)propyl)-2-(1,3-dioxo-6-(piperidin-1-yl)-1H-benzo[de]isoquinolin-2(3H)-yl)acetamide
N1-(7-chloroquinolin-4-yl)-N6-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)hexane-1,6-diamine
PfCRT-VMO
Photoaffinity labeling, suggested target
Primaquine
Promethazine
Quinacrine
Quinazoline
Quinine
qunidine
Saquinavir
Verapamil
W7
X-ray crystal structure, suggested target