You can find more information about
PF3D7_0934800-Protein kinase A
using the following links:
PlasmoDB - the Plasmodium genome resource
The TDR Targets Database
Subcellular Localization
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Affecting Drugs
Drug Name
PubMed Articles (year of publication)
(4aR,6R,7R,7aS)-6-(6-amino-2-chloro-purin-9-yl)-2-hydroxy-2-thioxo-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-ol
Disrupting the Allosteric Interaction between the Plasmodium falciparum cAMP-dependent Kinase and Its Regulatory Subunit(2016)
(4aR,6R,7R,7aS)-6-(6-amino-8-bromo-purin-9-yl)-2-hydroxy-2-thioxo-4a,6,7,7a-tetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-ol
Disrupting the Allosteric Interaction between the Plasmodium falciparum cAMP-dependent Kinase and Its Regulatory Subunit(2016)
1-(tert-Butylamino)-3-methylisoquinoline-4-carbonitrile
Exploration of 3-methylisoquinoline-4-carbonitriles as protein kinase A inhibitors of Plasmodium falciparum(2016)
3-Methyl-1-(pentylamino)isoquinoline-4-carbonitrile
Exploration of 3-methylisoquinoline-4-carbonitriles as protein kinase A inhibitors of Plasmodium falciparum(2016)
6-bz-camp
Cyclic AMP and calcium interplay as second messengers in melatonin-dependent regulation of Plasmodium falciparum cell cycle(2005)
Enzymatic properties, suggested target
Expression and biochemical characterization of the Plasmodium falciparum protein kinase A catalytic subunit(2009)
H89
The H89 cAMP-dependent protein kinase inhibitor blocks Plasmodium falciparum development in infected erythrocytes(2001)
H-89
Protein Kinase A Is Essential for Invasion of Plasmodium falciparum into Human Erythrocytes(2019)
Ibmx
Cyclic AMP and calcium interplay as second messengers in melatonin-dependent regulation of Plasmodium falciparum cell cycle(2005)
N-[2-[[3-(4-bromophenyl)-2-propenyl]amino]ethyl]-5-isoquinolinesulfonamide
Antimalarial activity of novel 4-cyano-3-methylisoquinoline inhibitors against Plasmodium falciparum: design, synthesis and biological evaluation(2016)