Malaria Parasite Metabolic Pathways
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Drug
Mode of action
Synergy between antimalarial compounds
Synergy between antimalarial compounds
Mason DJ, Eastman RT, Lewis RPI, Stott IP, Guha R, Bender A. Using Machine Learning to Predict Synergistic Antimalarial Compound Combinations With Novel Structures. Front Pharmacol. 2018 Oct 2;9:1096. PubMed PMID: 30333748
Drug A
Drug B
Synergy Value
Synergy
Tacrolimus
Hydroxyzine Pamoate
0.88491
Synergistic
Paroxetine
Guanethidine Sulfate
0.8885
Synergistic
Guanethidine Sulfate
Thioridazine
0.89458
Synergistic
Virginiamycin S1
Tacrolimus
0.90496
Synergistic
Fulvestrant
Tacrolimus
0.90815
Synergistic
Sorafenib tosylate
Hydroxyzine Pamoate
0.91655
Synergistic
CK2 Inhibitor II
Paroxetine
0.91702
Synergistic
Ingenol 3-Angelate
Tacrolimus
0.91714
Synergistic
Fulvestrant
Megesterol acetate
0.91775
Synergistic
Megesterol acetate
Hydroxyzine Pamoate
0.91987
Synergistic
Hydroxyzine Pamoate
Guanethidine Sulfate
0.92024
Synergistic
Dihydroergotamine
Thioridazine
0.92439
Synergistic
Apicidin
Dihydroergotamine
0.92439
Synergistic
Guanethidine Sulfate
Trifluoperazine 2HCl
0.92566
Synergistic
Virginiamycin S1
Sorafenib tosylate
0.92603
Synergistic
Thioridazine
Trifluoperazine 2HCl
0.92634
Synergistic
Tacrolimus
Dihydroergotamine
0.92932
Synergistic
Hydroxyzine Pamoate
Dihydroergotamine
0.93164
Synergistic
Tacrolimus
Thioridazine
0.93235
Synergistic
Sorafenib tosylate
Fulvestrant
0.9332
Synergistic
Sorafenib tosylate
Thioridazine
0.93472
Synergistic
PI 828
Guanethidine Sulfate
0.93511
Synergistic
Tacrolimus
Trifluoperazine 2HCl
0.93579
Synergistic
Dihydroergotamine
Guanethidine Sulfate
0.93655
Synergistic
Ingenol 3-Angelate
Apicidin
0.93669
Synergistic
Sorafenib tosylate
Trifluoperazine 2HCl
0.93743
Synergistic
Virginiamycin S1
Paroxetine
0.93784
Synergistic
PDK1 Inhibitor
Hydroxyzine Pamoate
0.93804
Synergistic
Ingenol 3-Angelate
Sorafenib tosylate
0.93804
Synergistic
Virginiamycin S1
Dihydroergotamine
0.94116
Synergistic
Apicidin
Tacrolimus
0.94229
Synergistic
Tacrolimus
Paroxetine
0.94421
Synergistic
Chromomycin A3
Fulvestrant
0.94734
Synergistic
Virginiamycin S1
Raloxifene HCl
0.9479
Synergistic
Dihydroergotamine
Raloxifene HCl
0.94993
Synergistic
Wortmannin
Guanethidine Sulfate
0.95002
Synergistic
Sorafenib tosylate
Dihydroergotamine
0.95076
Synergistic
CK2 Inhibitor II
Megesterol acetate
0.95166
Synergistic
Fulvestrant
Raloxifene HCl
0.95234
Synergistic
Apicidin
Hydroxyzine Pamoate
0.95242
Synergistic
Sorafenib tosylate
Tacrolimus
0.95245
Synergistic
Virginiamycin S1
Megesterol acetate
0.95361
Synergistic
Fulvestrant
Thioridazine
0.95437
Synergistic
Thioridazine
Raloxifene HCl
0.95586
Synergistic
Raloxifene HCl
Trifluoperazine 2HCl
0.95588
Synergistic
Apicidin
Virginiamycin S1
0.95673
Synergistic
Guanethidine Sulfate
Raloxifene HCl
0.95798
Synergistic
Dihydroergotamine
Trifluoperazine 2HCl
0.9584
Synergistic
PDK1 Inhibitor
Apicidin
0.95903
Synergistic
PDK1 Inhibitor
Raloxifene HCl
0.96025
Additive
Ingenol 3-Angelate
Thioridazine
0.96066
Additive
PI 828
Hydroxyzine Pamoate
0.96075
Additive
Megesterol acetate
Trifluoperazine 2HCl
0.96104
Additive
Fulvestrant
Trifluoperazine 2HCl
0.96165
Additive
PDK1 Inhibitor
Thioridazine
0.96179
Additive
Ciprofloxacin
Trifluoperazine 2HCl
0.96182
Additive
Fulvestrant
Hydroxyzine Pamoate
0.96243
Additive
Ingenol 3-Angelate
Dihydroergotamine
0.9627
Additive
Megesterol acetate
Dihydroergotamine
0.96328
Additive
PDK1 Inhibitor
Tacrolimus
0.96399
Additive
Chromomycin A3
CK2 Inhibitor II
0.96443
Additive
Tacrolimus
Raloxifene HCl
0.96447
Additive
Ingenol 3-Angelate
Megesterol acetate
0.9655
Additive
Wortmannin
Hydroxyzine Pamoate
0.96564
Additive
Paroxetine
Hydroxyzine Pamoate
0.96567
Additive
Tacrolimus
Guanethidine Sulfate
0.9658
Additive
Megesterol acetate
Guanethidine Sulfate
0.96597
Additive
PDK1 Inhibitor
Fulvestrant
0.96597
Additive
Apicidin
Trifluoperazine 2HCl
0.96638
Additive
PI 828
Fulvestrant
0.96743
Additive
Apicidin
Thioridazine
0.96757
Additive
CK2 Inhibitor II
Thioridazine
0.96758
Additive
Ingenol 3-Angelate
JX-401
0.96768
Additive
Megesterol acetate
Raloxifene HCl
0.96856
Additive
PI 828
Trifluoperazine 2HCl
0.96885
Additive
Ingenol 3-Angelate
Paroxetine
0.97085
Additive
Ingenol 3-Angelate
Trifluoperazine 2HCl
0.97151
Additive
Fulvestrant
Paroxetine
0.97212
Additive
Virginiamycin S1
Hydroxyzine Pamoate
0.97385
Additive
Ingenol 3-Angelate
Raloxifene HCl
0.97529
Additive
Sorafenib tosylate
Paroxetine
0.97529
Additive
Apicidin
Raloxifene HCl
0.97561
Additive
JX-401
Guanethidine Sulfate
0.97651
Additive
Apicidin
Fulvestrant
0.97666
Additive
Ciprofloxacin
Thioridazine
0.97672
Additive
Paroxetine
Raloxifene HCl
0.97686
Additive
Wortmannin
Trifluoperazine 2HCl
0.9781
Additive
PDK1 Inhibitor
Guanethidine Sulfate
0.9783
Additive
Chromomycin A3
Hydroxyzine Pamoate
0.97876
Additive
PDK1 Inhibitor
Trifluoperazine 2HCl
0.97983
Additive
Fulvestrant
Dihydroergotamine
0.98015
Additive
Chromomycin A3
Dihydroergotamine
0.98019
Additive
Sorafenib tosylate
Raloxifene HCl
0.98038
Additive
PDK1 Inhibitor
Virginiamycin S1
0.98077
Additive
PDK1 Inhibitor
Paroxetine
0.98123
Additive
JX-401
Trifluoperazine 2HCl
0.98136
Additive
Ingenol 3-Angelate
Wortmannin
0.98335
Additive
Apicidin
JX-401
0.9835
Additive
Chromomycin A3
Virginiamycin S1
0.98368
Additive
Virginiamycin S1
Trifluoperazine 2HCl
0.98375
Additive
Hydroxyzine Pamoate
Raloxifene HCl
0.98438
Additive
Tacrolimus
Megesterol acetate
0.98521
Additive
Paroxetine
Trifluoperazine 2HCl
0.98678
Additive
Chromomycin A3
Tacrolimus
0.98696
Additive
JX-401
Hydroxyzine Pamoate
0.98738
Additive
Virginiamycin S1
Guanethidine Sulfate
0.9875
Additive
CK2 Inhibitor II
Dihydroergotamine
0.98759
Additive
Paroxetine
Dihydroergotamine
0.98816
Additive
Hydroxyzine Pamoate
Ciprofloxacin
0.98861
Additive
Megesterol acetate
Thioridazine
0.98926
Additive
JX-401
Dihydroergotamine
0.98991
Additive
Chromomycin A3
Thioridazine
0.99086
Additive
PI 828
Ingenol 3-Angelate
0.99093
Additive
PI 828
Dihydroergotamine
0.99255
Additive
JX-401
Raloxifene
0.9927
Additive
Sorafenib tosylate
Ciprofloxacin
0.99293
Additive
JX-401
Thioridazine
0.99314
Additive
PI 828
Thioridazine
0.99365
Additive
PI 828
Virginiamycin S1
0.9941
Additive
Hydroxyzine Pamoate
Thioridazine
0.99462
Additive
Apicidin
Wortmannin
0.99463
Additive
Fulvestrant
Ciprofloxacin
0.99639
Additive
PDK1 Inhibitor
Dihydroergotamine
0.99678
Additive
PI 828
Apicidin
0.99678
Additive
PI 828
Raloxifene HCl
0.99688
Additive
Apicidin
Guanethidine Sulfate
0.99719
Additive
Virginiamycin S1
Wortmannin
0.99722
Additive
Apicidin
Paroxetine
0.99736
Additive
Sorafenib tosylate
Megesterol acetate
0.99739
Additive
PDK1 Inhibitor
Sorafenib tosylate
0.99742
Additive
Ciprofloxacin
Guanethidine Sulfate
0.99747
Additive
Ingenol 3-Angelate
Chromomycin A3
0.99764
Additive
Fulvestrant
Wortmannin
0.99843
Additive
Chromomycin A3
JX-401
0.99852
Additive
Wortmannin
Megesterol acetate
0.99891
Additive
Paroxetine
Thioridazine
0.99941
Additive
JX-401
Tacrolimus
0.99976
Additive
Ciprofloxacin
Raloxifene HCl
1.00049
Additive
Fulvestrant
Guanethidine Sulfate
1.00137
Additive
Wortmannin
Raloxifene HCl
1.00176
Additive
Hydroxyzine Pamoate
Trifluoperazine 2HCl
1.00225
Additive
Megesterol acetate
Ciprofloxacin
1.00238
Additive
Paroxetine
Megesterol acetate
1.00306
Additive
Chromomycin A3
Sorafenib tosylate
1.0036
Additive
Chromomycin A3
Trifluoperazine 2HCl
1.00415
Additive
Apicidin
Megesterol acetate
1.00437
Additive
CK2 Inhibitor II
Hydroxyzine Pamoate
1.00469
Additive
PI 828
Paroxetine
1.00562
Additive
JX-401
Sorafenib tosylate
1.00563
Additive
Fulvestrant
CK2 Inhibitor II
1.00779
Additive
Chromomycin A3
Megesterol acetate
1.00967
Additive
Apicidin
Sorafenib tosylate
1.01
Additive
Chromomycin A3
Wortmannin
1.01073
Additive
Chromomycin A3
Paroxetine
1.01104
Additive
Virginiamycin S1
Ciprofloxacin
1.01138
Additive
Ingenol 3-Angelate
Virginiamycin S1
1.0116
Additive
Sorafenib tosylate
CK2 Inhibitor II
1.01161
Additive
CK2 Inhibitor II
Raloxifene HCl
1.01212
Additive
JX-401
Paroxetine
1.01261
Additive
Ingenol 3-Angelate
Guanethidine Sulfate
1.0136
Additive
Apicidin
Chromomycin A3
1.01366
Additive
PI 828
Tacrolimus
1.01372
Additive
Ingenol 3-Angelate
Fulvestrant
1.01429
Additive
Sorafenib tosylate
Wortmannin
1.01455
Additive
PDK1 Inhibitor
Ingenol 3-Angelate
1.01487
Additive
PDK1 Inhibitor
Megesterol acetate
1.01633
Additive
Virginiamycin S1
Fulvestrant
1.01641
Additive
JX-401
Megesterol acetate
1.01672
Additive
Chromomycin A3
Guanethidine Sulfate
1.01731
Additive
PI 828
Sorafenib tosylate
1.01773
Additive
Chromomycin A3
Raloxifene HCl
1.01903
Additive
Ingenol 3-Angelate
Hydroxyzine Pamoate
1.02146
Additive
Sorafenib
Guanethidine Sulfate
1.02239
Additive
Tacrolimus
CK2 Inhibitor II
1.02297
Additive
CK2 Inhibitor II
Trifluoperazine 2HCl
1.02453
Additive
Ingenol 3-Angelate
Ciprofloxacin
1.02465
Additive
Wortmannin
Thioridazine
1.03026
Additive
PDK1 Inhibitor
Chromomycin A3
1.03147
Additive
JX-401
Fulvestrant
1.03301
Additive
Tacrolimus
Ciprofloxacin
1.03677
Additive
Virginiamycin S1
CK2 Inhibitor II
1.03816
Additive
PI 828
Chromomycin A3
1.03831
Additive
Apicidin
CK2 Inhibitor II
1.03892
Additive
Wortmannin
Dihydroergotamine
1.08384
Antagonistic
Wortmannin
Tacrolimus
1.09785
Antagonistic
Online articles related to Synergy between antimalarial compounds retrieved from PubMed
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